Bioorganic and Medicinal Chemistry, 0968-0896

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  1. 2018
  2. Novel multi-target compounds in the quest for new chemotherapies against Alzheimer's disease: An experimental and theoretical study

    Martínez, A., Zahran, M., Gomez, M., Cooper, C., Guevara, J., Erik Ekengard, Ebbe Nordlander, Alcendor, R. & Hambleton, S., 2018 Sep 15, In : Bioorganic and Medicinal Chemistry. 26, 17, p. 4823-4840 18 p.

    Research output: Contribution to journalArticle

  3. 2017
  4. Improved molecular recognition of Carbonic Anhydrase IX by polypeptide conjugation to acetazolamide

    Yang, J., Katarina Koruza, Zoë Fisher, Wolfgang Knecht & Baltzer, L., 2017 Oct, In : Bioorganic and Medicinal Chemistry. 25, 20, p. 5838-5848

    Research output: Contribution to journalArticle

  5. Cystatin C peptidomimetic derivative with antimicrobial properties as a potential compound against wound infections

    Pikuła, M., Smuzyńska, M., Krzystyniak, A., Zieliński, M., Langa, P., Deptuła, M., Schumacher, A., Łata, J., Cichorek, M., Anders Grubb, Trzonkowski, P., Kasprzykowski, F. & Rodziewicz-Motowidło, S., 2017 Feb 15, In : Bioorganic and Medicinal Chemistry. 25, 4, p. 1431-1439 9 p.

    Research output: Contribution to journalArticle

  6. 2013
  7. Synthesis and biology of oligoethylene glycol linked naphthoxylosides.

    Thorsheim, K., Persson, A., Johnsson, R., Löfgren, J., Katrin Mani & Ulf Ellervik, 2013, In : Bioorganic & Medicinal Chemistry. 21, 11, p. 3310-3317

    Research output: Contribution to journalArticle

  8. 2011
  9. Synthesis, conformation and biology of naphthoxylosides.

    Siegbahn, A., Aili, U., Ochocinska, A., Olofsson, M., Rönnols, J., Katrin Mani, Widmalm, G. & Ellervik, U., 2011, In : Bioorganic & Medicinal Chemistry. 19, p. 4114-4126

    Research output: Contribution to journalArticle

  10. Triazoloquinazolinediones as novel high affinity ligands for the benzodiazepine site of GABA(A) receptors.

    Nilsson, J., Ritha Gidlöf, Nielsen, E. Ø., Liljefors, T., Nielsen, M. & Olov Sterner, 2011, In : Bioorganic & Medicinal Chemistry. 19, 1, p. 111-121

    Research output: Contribution to journalArticle

  11. 2010
  12. 1H-1,2,3-Triazol-1-yl thiodigalactoside derivatives as high affinity galectin-3 inhibitors

    Salameh, B. A., Cumpstey, I., Sundin, A., Hakon Leffler & Ulf Nilsson, 2010, In : Bioorganic & Medicinal Chemistry. 18, 14, p. 5367-5378

    Research output: Contribution to journalArticle

  13. In vitro TRPV1 activity of piperine derived amides

    Andres Correa, E., Högestätt, E., Olov Sterner, Echeverri, F. & Peter Zygmunt, 2010, In : Bioorganic & Medicinal Chemistry. 18, 9, p. 3299-3306

    Research output: Contribution to journalArticle

  14. Photolabile ubiquinone analogues for identification and characterization of quinone binding sites in proteins.

    Pei, Z., Gustavsson, T., Roth, R., Torbjörn Frejd & Hägerhäll, C., 2010, In : Bioorganic & Medicinal Chemistry. 18, p. 3457-3466

    Research output: Contribution to journalArticle

  15. 2009
  16. Synthesis and biological evaluation of reversible inhibitors of IdeS, a bacterial cysteine protease and virulence determinant

    Berggren, K., Johansson, B., Fex, T., Kihlberg, J., Lars Björck & Luthman, K., 2009, In : Bioorganic & Medicinal Chemistry. 17, 9, p. 3463-3470

    Research output: Contribution to journalArticle

  17. 2008
  18. Affinity of 3-acyl substituted 4-quinolones at the benzodiazepine site of GABAA receptors.

    Lager, E., Nilsson, J., Østergaard Nielsen, E., Nielsen, M., Liljefors, T. & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry. 16, 14, p. 6936-6948

    Research output: Contribution to journalArticle

  19. Bioactive alkenylphenols from Piper obliquum.

    Valdivia, C., Marquez, N., Eriksson, J., Vilaseca, A., Muñoz, E. & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry. 16, 7, p. 4120-4126

    Research output: Contribution to journalArticle

  20. Imidazo[1,2-a]pyridine derivatives as inhibitors of TNF-alpha expression in T cells

    Rether, J., Erkel, G., Anke, T., Eriksson Bajtner, J. & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry. 16, 3, p. 1236-1241

    Research output: Contribution to journalArticle

  21. SAR studies of capsazepinoid bronchodilators 3: The thiourea part (coupling region) and the 2-(4-chlorophenyl)ethyl moiety (C-region).

    Berglund, M., Dalence, M., Skogvall, S. & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry. 16, 5, p. 2529-2540

    Research output: Contribution to journalArticle

  22. SAR studies of capsazepinoid bronchodilators. Part 1: The importance of the catechol moiety and aspects of the B-ring structure.

    Dalence, M., Berglund, M., Skogvall, S. & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry. 16, 5, p. 2499-2512

    Research output: Contribution to journalArticle

  23. SAR studies of capsazepinoid bronchodilators. Part 2: Chlorination and catechol replacement in the A-ring.

    Berglund, M., Dalence, M., Skogvall, S. & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry. 16, 5, p. 2513-2528

    Research output: Contribution to journalArticle

  24. Synthesis of glutamic acid analogs as potent inhibitors of leukotriene A(4) hydrolase

    Kirkland, T. A., Adler, M., Bauman, J. G., Chen, M., Haeggstrom, J. Z., King, B., Kochanny, M. J., Liang, A. M., Mendoza, L., Phillips, G. B., Marjolein Thunnissen, Trinh, L., Whitlow, M., Ye, B., Ye, H., Parkinson, J. & Guilford, W. J., 2008, In : Bioorganic & Medicinal Chemistry. 16, 9, p. 4963-4983

    Research output: Contribution to journalArticle

  25. 2007
  26. Construction of polyamine-modified uridine and adenosine derivatives-evaluation of DNA binding capacity and cytotoxicity in vitro

    Ghatnekar, J., Hägerlöf, M., Stina Oredsson, Alm, K., Sofi Elmroth & Persson, T., 2007, In : Bioorganic & Medicinal Chemistry. 15, 23, p. 7426-7433

    Research output: Contribution to journalArticle

  27. Effects of oxygen-sulfur substitution on glycosaminoglycan-priming naphthoxylosides.

    Jacobsson, M., Katrin Mani & Ulf Ellervik, 2007, In : Bioorganic & Medicinal Chemistry. 15, 15, p. 5283-5299

    Research output: Contribution to journalArticle

  28. Synthesis and biology of bis-xylosylated dihydroxynaphthalenes.

    Johnsson, R., Katrin Mani & Ulf Ellervik, 2007, In : Bioorganic & Medicinal Chemistry. 15, 8, p. 2868-2877

    Research output: Contribution to journalArticle

  29. 2006
  30. Design, synthesis, and biological evaluation of combretastatin nitrogen-containing derivatives as inhibitors of tubulin assembly and vascular disrupting agents

    Monk, KA., Siles, R., Hadimani, MB., Mugabe, BE., Ackley, JF., Studerus, SW., Edvardsen, K., Trawick, ML., Garner, CM., Rhodes, MR., Pettit, GR. & Pinney, KG., 2006, In : Bioorganic & Medicinal Chemistry. 14, 9, p. 3231-3244

    Research output: Contribution to journalArticle

  31. Side-chain and backbone amide bond requirements for glycopeptide stimulation of T-cells obtained in a mouse model for rheumatoid arthritis

    Holm, L., Bockermann, R., Wellner, E., Bäcklund, J., Holmdahl, R. & Kihlberg, J., 2006, In : Bioorganic & Medicinal Chemistry. 14, 17, p. 5921-5932

    Research output: Contribution to journalArticle

  32. Synthesis of aromatic C-xylosides by position inversion of glucose

    Malmberg, J., Katrin Mani, Säwén, E., Wiren, A. & Ulf Ellervik, 2006, In : Bioorganic & Medicinal Chemistry. 14, 19, p. 6659-6665

    Research output: Contribution to journalArticle

  33. Thioureido N-acetyllactosamine derivatives as potent galectin-7 and 9N inhibitors

    Salameh, B., Sundin, A., Hakon Leffler & Ulf Nilsson, 2006, In : Bioorganic & Medicinal Chemistry. 14, 4, p. 1215-1220

    Research output: Contribution to journalArticle

  34. 2005
  35. Identification of the minimal glycopeptide core recognized by T cells in a model for rheumatoid arthritis

    Holm, L., Kjellen, P., Holmdahl, R. & Kihlberg, J., 2005, In : Bioorganic & Medicinal Chemistry. 13, 2, p. 473-482

    Research output: Contribution to journalArticle

  36. Tridemethylisovelleral, a potent cytotoxic agent

    Aujard, I., Röme, D., Arzel, E., Johansson, M. H., de Vos, D. & Olov Sterner, 2005, In : Bioorganic & Medicinal Chemistry. 13, 22, p. 6145-6150

    Research output: Contribution to journalArticle

  37. 2003
  38. Quantitative studies of the binding of the class II PapG adhesin from uropathogenic Escherichia coli to oligosaccharides.

    Larsson, A., Ohlsson, J., Dodson, K. W., Hultgren, S. J., Ulf Nilsson & Kihlberg, J., 2003, In : Bioorganic & Medicinal Chemistry. 11, 10, p. 2255-2261

    Research output: Contribution to journalArticle

  39. Role of the galactosyl moiety of collagen glycopeptides for T-cell stimulation in a model for rheumatoid arthritis

    Holm, B., Baquer, SM., Holm, L., Holmdahl, R. & Kihlberg, J., 2003, In : Bioorganic & Medicinal Chemistry. 11, 18, p. 3981-3987

    Research output: Contribution to journalArticle

  40. 1996
  41. Synthesis of 2'-Deoxyuridine 5'-(α,β-Imido)triphosphate: A Substrate Analogue and Potent Inhibitor of dUTPase

    Persson, T., Larsson, G. & Nyman, P-O., 1996, In : Bioorganic & Medicinal Chemistry. 4, 4, p. 553-556

    Research output: Contribution to journalArticle