Bioorganic and Medicinal Chemistry, 0968-0896

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  1. 1H-1,2,3-Triazol-1-yl thiodigalactoside derivatives as high affinity galectin-3 inhibitors

    Salameh, B. A., Cumpstey, I., Sundin, A., Hakon Leffler & Ulf Nilsson, 2010, In : Bioorganic & Medicinal Chemistry. 18, 14, p. 5367-5378

    Research output: Contribution to journalArticle

  2. Affinity of 3-acyl substituted 4-quinolones at the benzodiazepine site of GABAA receptors.

    Lager, E., Nilsson, J., Østergaard Nielsen, E., Nielsen, M., Liljefors, T. & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry. 16, 14, p. 6936-6948

    Research output: Contribution to journalArticle

  3. Bioactive alkenylphenols from Piper obliquum.

    Valdivia, C., Marquez, N., Eriksson, J., Vilaseca, A., Muñoz, E. & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry. 16, 7, p. 4120-4126

    Research output: Contribution to journalArticle

  4. Construction of polyamine-modified uridine and adenosine derivatives-evaluation of DNA binding capacity and cytotoxicity in vitro

    Ghatnekar, J., Hägerlöf, M., Stina Oredsson, Alm, K., Sofi Elmroth & Persson, T., 2007, In : Bioorganic & Medicinal Chemistry. 15, 23, p. 7426-7433

    Research output: Contribution to journalArticle

  5. Cystatin C peptidomimetic derivative with antimicrobial properties as a potential compound against wound infections

    Pikuła, M., Smuzyńska, M., Krzystyniak, A., Zieliński, M., Langa, P., Deptuła, M., Schumacher, A., Łata, J., Cichorek, M., Anders Grubb, Trzonkowski, P., Kasprzykowski, F. & Rodziewicz-Motowidło, S., 2017 Feb 15, In : Bioorganic and Medicinal Chemistry. 25, 4, p. 1431-1439 9 p.

    Research output: Contribution to journalArticle

  6. Design, synthesis, and biological evaluation of combretastatin nitrogen-containing derivatives as inhibitors of tubulin assembly and vascular disrupting agents

    Monk, KA., Siles, R., Hadimani, MB., Mugabe, BE., Ackley, JF., Studerus, SW., Edvardsen, K., Trawick, ML., Garner, CM., Rhodes, MR., Pettit, GR. & Pinney, KG., 2006, In : Bioorganic & Medicinal Chemistry. 14, 9, p. 3231-3244

    Research output: Contribution to journalArticle

  7. Effects of oxygen-sulfur substitution on glycosaminoglycan-priming naphthoxylosides.

    Jacobsson, M., Katrin Mani & Ulf Ellervik, 2007, In : Bioorganic & Medicinal Chemistry. 15, 15, p. 5283-5299

    Research output: Contribution to journalArticle

  8. Identification of the minimal glycopeptide core recognized by T cells in a model for rheumatoid arthritis

    Holm, L., Kjellen, P., Holmdahl, R. & Kihlberg, J., 2005, In : Bioorganic & Medicinal Chemistry. 13, 2, p. 473-482

    Research output: Contribution to journalArticle

  9. Imidazo[1,2-a]pyridine derivatives as inhibitors of TNF-alpha expression in T cells

    Rether, J., Erkel, G., Anke, T., Eriksson Bajtner, J. & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry. 16, 3, p. 1236-1241

    Research output: Contribution to journalArticle

  10. Improved molecular recognition of Carbonic Anhydrase IX by polypeptide conjugation to acetazolamide

    Yang, J., Katarina Koruza, Zoë Fisher, Wolfgang Knecht & Baltzer, L., 2017 Oct, In : Bioorganic and Medicinal Chemistry. 25, 20, p. 5838-5848

    Research output: Contribution to journalArticle

  11. In vitro TRPV1 activity of piperine derived amides

    Andres Correa, E., Högestätt, E., Olov Sterner, Echeverri, F. & Peter Zygmunt, 2010, In : Bioorganic & Medicinal Chemistry. 18, 9, p. 3299-3306

    Research output: Contribution to journalArticle

  12. Isochromanone-based urotensin-II receptor agonists

    Lehmann, F., Currier, E. A., Roger Olsson, Hacksell, U. & Luthman, K., 2005 Apr 15, In : Bioorganic and Medicinal Chemistry. 13, 8, p. 3057-3068 12 p.

    Research output: Contribution to journalArticle

  13. Novel and potent small-molecule urotensin II receptor agonists

    Lehmann, F., Currier, E. A., Clemons, B., Hansen, L. K., Roger Olsson, Hacksell, U. & Luthman, K., 2009 Jul 1, In : Bioorganic and Medicinal Chemistry. 17, 13, p. 4657-4665

    Research output: Contribution to journalArticle

  14. Novel multi-target compounds in the quest for new chemotherapies against Alzheimer's disease: An experimental and theoretical study

    Martínez, A., Zahran, M., Gomez, M., Cooper, C., Guevara, J., Ekengard, E., Ebbe Nordlander, Alcendor, R. & Hambleton, S., 2018 Sep 15, In : Bioorganic and Medicinal Chemistry. 26, 17, p. 4823-4840 18 p.

    Research output: Contribution to journalArticle

  15. Optimization of isochromanone based urotensin II receptor agonists

    Lehmann, F., Currier, E. A., Roger Olsson, Ma, J. N., Burstein, E. S., Hacksell, U. & Luthman, K., 2010 May 31, In : Bioorganic and Medicinal Chemistry. 18, 13, p. 4844-4854 11 p.

    Research output: Contribution to journalArticle

  16. Photolabile ubiquinone analogues for identification and characterization of quinone binding sites in proteins.

    Pei, Z., Gustavsson, T., Roth, R., Torbjörn Frejd & Hägerhäll, C., 2010, In : Bioorganic & Medicinal Chemistry. 18, p. 3457-3466

    Research output: Contribution to journalArticle

  17. Quantitative studies of the binding of the class II PapG adhesin from uropathogenic Escherichia coli to oligosaccharides.

    Larsson, A., Ohlsson, J., Dodson, K. W., Hultgren, S. J., Ulf Nilsson & Kihlberg, J., 2003, In : Bioorganic & Medicinal Chemistry. 11, 10, p. 2255-2261

    Research output: Contribution to journalArticle

  18. Reaction medium engineering in enzymatic peptide fragment condensation: Synthesis of eledoisin and LH-RH

    Björup, P., Torres, J. L., Patrick Adlercreutz & Clapés, P., 1998 Jul 1, In : Bioorganic and Medicinal Chemistry. 6, 7, p. 891-901 11 p.

    Research output: Contribution to journalArticle

  19. Role of the galactosyl moiety of collagen glycopeptides for T-cell stimulation in a model for rheumatoid arthritis

    Holm, B., Baquer, SM., Holm, L., Holmdahl, R. & Kihlberg, J., 2003, In : Bioorganic & Medicinal Chemistry. 11, 18, p. 3981-3987

    Research output: Contribution to journalArticle

  20. SAR studies of capsazepinoid bronchodilators 3: The thiourea part (coupling region) and the 2-(4-chlorophenyl)ethyl moiety (C-region).

    Berglund, M., Dalence, M., Skogvall, S. & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry. 16, 5, p. 2529-2540

    Research output: Contribution to journalArticle

  21. SAR studies of capsazepinoid bronchodilators. Part 1: The importance of the catechol moiety and aspects of the B-ring structure.

    Dalence, M., Berglund, M., Skogvall, S. & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry. 16, 5, p. 2499-2512

    Research output: Contribution to journalArticle

  22. SAR studies of capsazepinoid bronchodilators. Part 2: Chlorination and catechol replacement in the A-ring.

    Berglund, M., Dalence, M., Skogvall, S. & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry. 16, 5, p. 2513-2528

    Research output: Contribution to journalArticle

  23. Side-chain and backbone amide bond requirements for glycopeptide stimulation of T-cells obtained in a mouse model for rheumatoid arthritis

    Holm, L., Bockermann, R., Wellner, E., Bäcklund, J., Holmdahl, R. & Kihlberg, J., 2006, In : Bioorganic & Medicinal Chemistry. 14, 17, p. 5921-5932

    Research output: Contribution to journalArticle

  24. Synthesis and biological evaluation of reversible inhibitors of IdeS, a bacterial cysteine protease and virulence determinant

    Berggren, K., Johansson, B., Fex, T., Kihlberg, J., Lars Björck & Luthman, K., 2009, In : Bioorganic & Medicinal Chemistry. 17, 9, p. 3463-3470

    Research output: Contribution to journalArticle

  25. Synthesis and biology of bis-xylosylated dihydroxynaphthalenes.

    Johnsson, R., Katrin Mani & Ulf Ellervik, 2007, In : Bioorganic & Medicinal Chemistry. 15, 8, p. 2868-2877

    Research output: Contribution to journalArticle

  26. Synthesis and biology of oligoethylene glycol linked naphthoxylosides.

    Thorsheim, K., Persson, A., Johnsson, R., Löfgren, J., Katrin Mani & Ulf Ellervik, 2013, In : Bioorganic & Medicinal Chemistry. 21, 11, p. 3310-3317

    Research output: Contribution to journalArticle

  27. Synthesis, conformation and biology of naphthoxylosides.

    Siegbahn, A., Aili, U., Ochocinska, A., Olofsson, M., Rönnols, J., Katrin Mani, Widmalm, G. & Ellervik, U., 2011, In : Bioorganic & Medicinal Chemistry. 19, p. 4114-4126

    Research output: Contribution to journalArticle

  28. Synthesis of 2'-Deoxyuridine 5'-(α,β-Imido)triphosphate: A Substrate Analogue and Potent Inhibitor of dUTPase

    Persson, T., Larsson, G. & Nyman, P-O., 1996, In : Bioorganic & Medicinal Chemistry. 4, 4, p. 553-556

    Research output: Contribution to journalArticle

  29. Synthesis of aromatic C-xylosides by position inversion of glucose

    Malmberg, J., Katrin Mani, Säwén, E., Wiren, A. & Ulf Ellervik, 2006, In : Bioorganic & Medicinal Chemistry. 14, 19, p. 6659-6665

    Research output: Contribution to journalArticle

  30. Synthesis of glutamic acid analogs as potent inhibitors of leukotriene A(4) hydrolase

    Kirkland, T. A., Adler, M., Bauman, J. G., Chen, M., Haeggstrom, J. Z., King, B., Kochanny, M. J., Liang, A. M., Mendoza, L., Phillips, G. B., Marjolein Thunnissen, Trinh, L., Whitlow, M., Ye, B., Ye, H., Parkinson, J. & Guilford, W. J., 2008, In : Bioorganic & Medicinal Chemistry. 16, 9, p. 4963-4983

    Research output: Contribution to journalArticle

  31. Synthetic polymers as solubilizing vehicles for enzymes in water-poor media

    Patrick Adlercreutz, Bo Matiasson & Otamiri, M., 1994 Jan 1, In : Bioorganic and Medicinal Chemistry. 2, 6, p. 529-533 5 p.

    Research output: Contribution to journalArticle

  32. Thioureido N-acetyllactosamine derivatives as potent galectin-7 and 9N inhibitors

    Salameh, B., Sundin, A., Hakon Leffler & Ulf Nilsson, 2006, In : Bioorganic & Medicinal Chemistry. 14, 4, p. 1215-1220

    Research output: Contribution to journalArticle

  33. Triazoloquinazolinediones as novel high affinity ligands for the benzodiazepine site of GABA(A) receptors.

    Nilsson, J., Ritha Gidlöf, Nielsen, E. Ø., Liljefors, T., Nielsen, M. & Olov Sterner, 2011, In : Bioorganic & Medicinal Chemistry. 19, 1, p. 111-121

    Research output: Contribution to journalArticle

  34. Tridemethylisovelleral, a potent cytotoxic agent

    Aujard, I., Röme, D., Arzel, E., Johansson, M. H., de Vos, D. & Olov Sterner, 2005, In : Bioorganic & Medicinal Chemistry. 13, 22, p. 6145-6150

    Research output: Contribution to journalArticle