Bioorganic and Medicinal Chemistry Letters, 0960-894X

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  1. 2016
  2. Reactivity of the glutathione species towards the reduction of ormaplatin (or tetraplatin)

    Jingran Dong, Shuying Huo, Shigang Shen, Jianzhong Xu, Tiesheng Shi & Lars Ivar Elding, 2016 Sep 1, In : Bioorganic and Medicinal Chemistry Letters. 26, 17, p. 4261-4266 6 p.

    Research output: Contribution to journalArticle

  3. 2014
  4. Bexarotene prodrugs: Targeting through cleavage by NQO1 (DT-diaphorase).

    Anja Schäfer, Ethan S Burstein & Roger Olsson, 2014, In : Bioorganic & Medicinal Chemistry Letters. 24, 8, p. 1944-1947

    Research output: Contribution to journalArticle

  5. HTS followed by NMR based counterscreening. Discovery and optimization of pyrimidones as reversible and competitive inhibitors of xanthine oxidase.

    Johan Evenäs, Fredrik Edfeldt, Matti Lepistö, Naila Svitacheva, Anna Synnergren, Britta Lundquist, Mia Gränse, Anna Rönnholm, Mikael Varga, John Wright, Min Wei, Sherrie Yue, Junfeng Wang, Chong Li, Xuan Li, Gang Chen, Yong Liao, Gang Lv, Ann Tjörnebo & Frank Narjes, 2014, In : Bioorganic & Medicinal Chemistry Letters. 24, 5, p. 1315-1321

    Research output: Contribution to journalArticle

  6. Synthesis and evaluation of iminocoumaryl and coumaryl derivatized glycosides as galectin antagonists.

    Vishal Kumar Rajput, Hakon Leffler, Ulf J Nilsson & Balaram Mukhopadhyay, 2014, In : Bioorganic & Medicinal Chemistry Letters. 24, 15, p. 3516-3520

    Research output: Contribution to journalArticle

  7. 2012
  8. Discovery of benzothiazole guanidines as novel inhibitors of thrombin and trypsin IV

    Michael Karle, Wolfgang Knecht & Yafeng Xue, 2012 Jul 15, In : Bioorganic & Medicinal Chemistry Letters. 22, 14, p. 4839-4843

    Research output: Contribution to journalArticle

  9. Discovery of 4-hydroxy-1,6-naphthyridine-3-carbonitrile derivatives as novel PDE10A inhibitors

    Udo Bauer, Fabrizio Giordanetto, Martin Bauer, Gavin O'Mahony, Kjell E Johansson, Wolfgang Knecht, Judith Hartleib-Geschwindner, Eva Töppner Carlsson & Cristofer Enroth, 2012 Mar 1, In : Bioorganic & Medicinal Chemistry Letters. 22, 5, p. 1944-1948

    Research output: Contribution to journalArticle

  10. 2011
  11. 3-Alkyl- and 3-amido-isothiazoloquinolin-4-ones as ligands for the benzodiazepine site of GABA(A) receptors.

    Jakob Nilsson, Elsebet Ostergaard Nielsen, Tommy Liljefors, Mogens Nielsen & Olov Sterner, 2011, In : Bioorganic & Medicinal Chemistry Letters.

    Research output: Contribution to journalArticle

  12. 2010
  13. Design and synthesis of macrocyclic indoles targeting blood coagulation cascade Factor XIa

    Stephen Hanessian, Andreas Larsson, Tomas Fex, Wolfgang Knecht & Niklas Blomberg, 2010 Dec 1, In : Bioorganic & Medicinal Chemistry Letters. 20, 23, p. 6925-6928

    Research output: Contribution to journalArticle

  14. Discovery of a class of calcium sensing receptor positive allosteric modulators; 1-(benzothiazol-2-yl)-1-phenylethanols

    Magnus Gustafsson, Jacob Jensen, Sine M. Bertozzi, Erika A. Currier, Jian Nong Ma, Ethan S. Burstein & Roger Olsson, 2010 Oct 1, In : Bioorganic and Medicinal Chemistry Letters. 20, 19, p. 5918-5921 4 p.

    Research output: Contribution to journalArticle

  15. 2009
  16. Discovery of non-peptidergic MrgX1 and MrgX2 receptor agonists and exploration of an initial SAR using solid-phase synthesis

    Leila Malik, Nicholas M. Kelly, Jian Nong Ma, Erika A. Currier, Ethan S. Burstein & Roger Olsson, 2009 Mar 15, In : Bioorganic and Medicinal Chemistry Letters. 19, 6, p. 1729-1732 4 p.

    Research output: Contribution to journalArticle

  17. Antiproliferative effects of peracetylated naphthoxylosides.

    Ulrika Aili, Mårten Jacobsson, Richard Johnsson, Katrin Mani & Ulf Ellervik, 2009, In : Bioorganic & Medicinal Chemistry Letters. 19, p. 1763-1766

    Research output: Contribution to journalArticle

  18. 2008
  19. Azaflavones compared to flavones as ligands to the benzodiazepine binding site of brain GABA(A) receptors.

    Jakob Nilsson, Elsebet Østergaard Nielsen, Tommy Liljefors, Mogens Nielsen & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry Letters. 18, 21, p. 5713-5716

    Research output: Contribution to journalArticle

  20. Protein subtype-targeting through ligand epimerization: talose-selectivity of galectin-4 and galectin-8.

    Christopher Öberg, Helen Blanchard, Hakon Leffler & Ulf Nilsson, 2008, In : Bioorganic & Medicinal Chemistry Letters. 18, 13, p. 3691-3694

    Research output: Contribution to journalArticle

  21. Xylose as a carrier for boron containing compounds.

    Mårten Jacobsson, Cecilia Winander, Katrin Mani & Ulf Ellervik, 2008, In : Bioorganic & Medicinal Chemistry Letters. 18, 7, p. 2451-2454

    Research output: Contribution to journalArticle

  22. 2007
  23. Evaluation of fluorescently labeled xylopyranosides as probes for proteoglycan biosynthesis

    Richard Johnsson, Katrin Mani & Ulf Ellervik, 2007, In : Bioorganic & Medicinal Chemistry Letters. 17, 8, p. 2338-2341

    Research output: Contribution to journalArticle

  24. 2005
  25. Synthesis of O-galactosyl aldoximes as potent LacNAc-mimetic galectin-3 inhibitors.

    Johan Tejler, Hakon Leffler & Ulf Nilsson, 2005, In : Bioorganic & Medicinal Chemistry Letters. 15, 9, p. 2343-2345

    Research output: Contribution to journalArticle

  26. 2003
  27. Synthesis, in vitro, and in vivo evaluation of phosphate ester derivatives of combretastatin A-4

    MB Hadimani, Jianyi Hua, MD Jonklaas, RJ Kessler, Yezhou Sheng, A Olivares, RP Tanpure, A Weiser, JX Zhang, Klaus Edvardsen, RR Kane & KG Pinney, 2003, In : Bioorganic & Medicinal Chemistry Letters. 13, 9, p. 1505-1508

    Research output: Contribution to journalArticle

  28. Xylylated dimers of putrescine and polyamines: influence of the polyamine backbone on spermidine transport inhibition

    Laurence Covassin, Michel Desjardins, Denis Soulet, Rene Charest-Gaudreault, Marie Audette & Richard Poulin, 2003, In : Bioorganic & Medicinal Chemistry Letters. 13, 19, p. 3267-3271

    Research output: Contribution to journalArticle

  29. 2000
  30. Multistep solution-phase parallel synthesis of spiperone analogues

    Henrik C. Hansen, Roger Olsson, Glenn Croston & Carl Magnus Andersson, 2000 Nov 6, In : Bioorganic and Medicinal Chemistry Letters. 10, 21, p. 2435-2439

    Research output: Contribution to journalArticle