Bioorganic and Medicinal Chemistry Letters, 0960-894X
Journal
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Reactivity of the glutathione species towards the reduction of ormaplatin (or tetraplatin)
Jingran Dong, Shuying Huo, Shigang Shen, Jianzhong Xu, Tiesheng Shi & Lars Ivar Elding, 2016 Sep 1, In : Bioorganic and Medicinal Chemistry Letters. 26, 17, p. 4261-4266 6 p.Research output: Contribution to journal › Article
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Synthesis and evaluation of iminocoumaryl and coumaryl derivatized glycosides as galectin antagonists.
Vishal Kumar Rajput, Hakon Leffler, Ulf J Nilsson & Balaram Mukhopadhyay, 2014, In : Bioorganic & Medicinal Chemistry Letters. 24, 15, p. 3516-3520Research output: Contribution to journal › Article
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Bexarotene prodrugs: Targeting through cleavage by NQO1 (DT-diaphorase).
Anja Schäfer, Ethan S Burstein & Roger Olsson, 2014, In : Bioorganic & Medicinal Chemistry Letters. 24, 8, p. 1944-1947Research output: Contribution to journal › Article
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HTS followed by NMR based counterscreening. Discovery and optimization of pyrimidones as reversible and competitive inhibitors of xanthine oxidase.
Johan Evenäs, Fredrik Edfeldt, Matti Lepistö, Naila Svitacheva, Anna Synnergren, Britta Lundquist, Mia Gränse, Anna Rönnholm, Mikael Varga, John Wright, Min Wei, Sherrie Yue, Junfeng Wang, Chong Li, Xuan Li, Gang Chen, Yong Liao, Gang Lv, Ann Tjörnebo & Frank Narjes, 2014, In : Bioorganic & Medicinal Chemistry Letters. 24, 5, p. 1315-1321Research output: Contribution to journal › Article
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Discovery of benzothiazole guanidines as novel inhibitors of thrombin and trypsin IV
Michael Karle, Wolfgang Knecht & Yafeng Xue, 2012 Jul 15, In : Bioorganic & Medicinal Chemistry Letters. 22, 14, p. 4839-4843Research output: Contribution to journal › Article
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Discovery of 4-hydroxy-1,6-naphthyridine-3-carbonitrile derivatives as novel PDE10A inhibitors
Udo Bauer, Fabrizio Giordanetto, Martin Bauer, Gavin O'Mahony, Kjell E Johansson, Wolfgang Knecht, Judith Hartleib-Geschwindner, Eva Töppner Carlsson & Cristofer Enroth, 2012 Mar 1, In : Bioorganic & Medicinal Chemistry Letters. 22, 5, p. 1944-1948Research output: Contribution to journal › Article
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3-Alkyl- and 3-amido-isothiazoloquinolin-4-ones as ligands for the benzodiazepine site of GABA(A) receptors.
Jakob Nilsson, Elsebet Ostergaard Nielsen, Tommy Liljefors, Mogens Nielsen & Olov Sterner, 2011, In : Bioorganic & Medicinal Chemistry Letters.Research output: Contribution to journal › Article
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Design and synthesis of macrocyclic indoles targeting blood coagulation cascade Factor XIa
Stephen Hanessian, Andreas Larsson, Tomas Fex, Wolfgang Knecht & Niklas Blomberg, 2010 Dec 1, In : Bioorganic & Medicinal Chemistry Letters. 20, 23, p. 6925-6928Research output: Contribution to journal › Article
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Discovery of a class of calcium sensing receptor positive allosteric modulators; 1-(benzothiazol-2-yl)-1-phenylethanols
Magnus Gustafsson, Jacob Jensen, Sine M. Bertozzi, Erika A. Currier, Jian Nong Ma, Ethan S. Burstein & Roger Olsson, 2010 Oct 1, In : Bioorganic and Medicinal Chemistry Letters. 20, 19, p. 5918-5921 4 p.Research output: Contribution to journal › Article
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Discovery of non-peptidergic MrgX1 and MrgX2 receptor agonists and exploration of an initial SAR using solid-phase synthesis
Leila Malik, Nicholas M. Kelly, Jian Nong Ma, Erika A. Currier, Ethan S. Burstein & Roger Olsson, 2009 Mar 15, In : Bioorganic and Medicinal Chemistry Letters. 19, 6, p. 1729-1732 4 p.Research output: Contribution to journal › Article
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Antiproliferative effects of peracetylated naphthoxylosides.
Ulrika Aili, Mårten Jacobsson, Richard Johnsson, Katrin Mani & Ulf Ellervik, 2009, In : Bioorganic & Medicinal Chemistry Letters. 19, p. 1763-1766Research output: Contribution to journal › Article
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Azaflavones compared to flavones as ligands to the benzodiazepine binding site of brain GABA(A) receptors.
Jakob Nilsson, Elsebet Østergaard Nielsen, Tommy Liljefors, Mogens Nielsen & Olov Sterner, 2008, In : Bioorganic & Medicinal Chemistry Letters. 18, 21, p. 5713-5716Research output: Contribution to journal › Article
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Xylose as a carrier for boron containing compounds.
Mårten Jacobsson, Cecilia Winander, Katrin Mani & Ulf Ellervik, 2008, In : Bioorganic & Medicinal Chemistry Letters. 18, 7, p. 2451-2454Research output: Contribution to journal › Article
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Protein subtype-targeting through ligand epimerization: talose-selectivity of galectin-4 and galectin-8.
Christopher Öberg, Helen Blanchard, Hakon Leffler & Ulf Nilsson, 2008, In : Bioorganic & Medicinal Chemistry Letters. 18, 13, p. 3691-3694Research output: Contribution to journal › Article
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Evaluation of fluorescently labeled xylopyranosides as probes for proteoglycan biosynthesis
Richard Johnsson, Katrin Mani & Ulf Ellervik, 2007, In : Bioorganic & Medicinal Chemistry Letters. 17, 8, p. 2338-2341Research output: Contribution to journal › Article
Synthesis of O-galactosyl aldoximes as potent LacNAc-mimetic galectin-3 inhibitors.
Johan Tejler, Hakon Leffler & Ulf Nilsson, 2005, In : Bioorganic & Medicinal Chemistry Letters. 15, 9, p. 2343-2345Research output: Contribution to journal › Article
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3-(1,2,3-Triazol-1-yl)-1-thio-galactosides as small, efficient, and hydrolytically stable inhibitors of galectin-3
Bader Salameh, Hakon Leffler & Ulf Nilsson, 2005, In : Bioorganic & Medicinal Chemistry Letters. 15, 14, p. 3344-3346Research output: Contribution to journal › Article
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Synthesis, in vitro, and in vivo evaluation of phosphate ester derivatives of combretastatin A-4
MB Hadimani, Jianyi Hua, MD Jonklaas, RJ Kessler, Yezhou Sheng, A Olivares, RP Tanpure, A Weiser, JX Zhang, Klaus Edvardsen, RR Kane & KG Pinney, 2003, In : Bioorganic & Medicinal Chemistry Letters. 13, 9, p. 1505-1508Research output: Contribution to journal › Article
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Xylylated dimers of putrescine and polyamines: influence of the polyamine backbone on spermidine transport inhibition
Laurence Covassin, Michel Desjardins, Denis Soulet, Rene Charest-Gaudreault, Marie Audette & Richard Poulin, 2003, In : Bioorganic & Medicinal Chemistry Letters. 13, 19, p. 3267-3271Research output: Contribution to journal › Article
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Multistep solution-phase parallel synthesis of spiperone analogues
Henrik C. Hansen, Roger Olsson, Glenn Croston & Carl Magnus Andersson, 2000 Nov 6, In : Bioorganic and Medicinal Chemistry Letters. 10, 21, p. 2435-2439Research output: Contribution to journal › Article