Design, synthesis, biological evaluation and X-ray structural studies of potent human dihydroorotate dehydrogenase inhibitors based on hydroxylated azole scaffolds

Stefano Sainas, Agnese C. Pippione, Marta Giorgis, Elisa Lupino, Parveen Goyal, Cristina Ramondetti, Barbara Buccinnà, Marco Piccinini, Rodolpho C. Braga, Carolina H. Andrade, Mikael Andersson, Ann Christin Moritzer, Rosmarie Friemann, Stefano Mensa, Salam Al-Karadaghi, Donatella Boschi, Marco L. Lolli

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Pharmacology, Toxicology and Pharmaceutical Science